GPER
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G protein-coupled estrogen receptor 1 (GPER), also known as G protein-coupled receptor 30 (GPR30), is a protein that in humans is encoded by the GPER gene. GPER binds to and is activated by the female sex hormone estradiol and is responsible for some of the rapid effects that estradiol has on cells.
G protein-coupled estrogen receptor 1 (GPER), also known as G protein-coupled receptor 30 (GPR30), is a protein that in humans is encoded by the GPER gene. GPER binds to and is activated by the female sex hormone estradiol and is responsible for some of the rapid effects that estradiol has on cells. ===Agonists=== 2-Methoxyestradiol 2,2',5'-PCB-4-OH Afimoxifene Aldosterone Atrazine Bisphenol A Daidzein DDT (p,p'-DDT, o',p'-DDE) Diarylpropionitrile (DPN) Equol Estradiol Ethynylestradiol Fulvestrant (ICI-182780)) G-1 Genistein GPER-L1 GPER-L2 Hydroxytyrosol Kepone LNS8801 Niacin Nicotinamide Nonylphenol Oleuropein Protocatechuic aldehyde Propylpyrazoletriol (PPT) Quercetin Raloxifene Resveratrol STX Tamoxifen Tectoridin ===Antagonists=== CCL18 Estriol G15 G36 MIBE ===Unknown=== Diethylstilbestrol Zearalenone ===Non-ligand=== 17α-Estradiol Estrone
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