NBUMP
≈ 1 min read
Names in other languages
No names in other languages are held for this entry yet.
Article bodies are English and are not machine-translated. A name in another language is not a translation of the article.
NBUMP is a highly selective 5-HT 1A receptor partial agonist (K i = 0.1 nM; IA = 40%) with an arylpiperazine structure. It is one of the highest affinity ligands for the 5-HT 1A receptor known. It displays 460- and 260-fold selectivity for 5-HT 1A over the α 1 -adrenergic and D 2 receptors, respectively.
NBUMP is a highly selective 5-HT 1A receptor partial agonist (K i = 0.1 nM; IA = 40%) with an arylpiperazine structure. It is one of the highest affinity ligands for the 5-HT 1A receptor known. It displays 460- and 260-fold selectivity for 5-HT 1A over the α 1 -adrenergic and D 2 receptors, respectively.
Text derived from https://en.wikipedia.org/w/index.php?oldid=1329172877 under CC BY-SA 4.0; modifications have been made.